selected publications
- The GR-LEDGF/p75-HSP27 Axis Contributes to Cross-Resistance Between Enzalutamide and Docetaxel in Prostate Cancer. Cells. 2025 Academic Article GET IT
- Chondrosarcoma: Multi-Targeting Therapeutic Effects of Doxorubicin, BEZ235, and the Small Molecule Aspartyl-Asparaginyl-β-hydroxylase Inhibitor SMI1182. Cancers. 2025 Academic Article GET IT
- Inhibition of Mitochondrial-Associated Protein MAGMAS Resensitizes Chemoresistant Prostate Cancer Cells to Docetaxel. Cancers. 2025 Academic Article GET IT
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Dual targeting of the mitochondrial Lon peptidase 1 and the chymotrypsin-like proteasome activity as a potential therapeutic strategy in malignant astrocytoma models.
Pharmacological research.
2025
Academic Article
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Times cited: 1 - Methionine Aminopeptidase 2 (MetAP2) Inhibitor BL6 Attenuates Inflammation in Cultured Microglia and in a Mouse Model of Alzheimer's Disease. Molecules (Basel, Switzerland). 2025 Academic Article GET IT
- Shroom3-Rock interaction and profibrotic function: Resolving mechanism of an intronic CKD risk allele. 2024 GET IT
- Preclinical assessment of MAGMAS inhibitor as a potential therapy for pediatric medulloblastoma. PloS one. 2024 Academic Article GET IT
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Targeting Krüppel-Like Factor 2 as a Novel Therapy for Glomerular Endothelial Cell Injury in Diabetic Kidney Disease.
Journal of the American Society of Nephrology : JASN.
2024
Academic Article
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Times cited: 2 -
Methionine aminopeptidases: Potential therapeutic target for microsporidia and other microbes.
The Journal of eukaryotic microbiology.
2024
Review
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Times cited: 5 -
HCK induces macrophage activation to promote renal inflammation and fibrosis via suppression of autophagy.
Nature communications.
2023
Academic Article
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Times cited: 64 -
Identification of new hit to lead magmas inhibitors as potential therapeutics for glioblastoma.
Bioorganic & medicinal chemistry letters.
2023
Academic Article
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Times cited: 1 -
Effects of retinoic acid receptor α modulators on developmental ethanol-induced neurodegeneration and neuroinflammation.
Frontiers in neuroscience.
2023
Academic Article
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Times cited: 1 -
Anti-inflammatory Action of BT75, a Novel RARα Agonist, in Cultured Microglia and in an Experimental Mouse Model of Alzheimer's Disease.
Neurochemical research.
2023
Academic Article
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Times cited: 11 -
Stimuli-Responsive Boron-Based Materials in Drug Delivery.
International journal of molecular sciences.
2023
Review
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Times cited: 38 -
Development of a New Methodology for Dearomative Borylation of Coumarins and Chromenes and Its Applications to Synthesize Boron-Containing Retinoids.
Molecules (Basel, Switzerland).
2023
Academic Article
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Times cited: 2 -
TYRO3 agonist as therapy for glomerular disease.
JCI insight.
2023
Academic Article
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Times cited: 11 -
New Boron Delivery Agents.
Cancer biotherapy & radiopharmaceuticals.
2022
Review
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Times cited: 29 -
A novel procedure for the synthesis of borylated quinolines and its application in the development of potential boron-based homeodomain interacting protein kinase 2 (HIPK2) inhibitors.
RSC advances.
2022
Academic Article
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Times cited: 5 - Tackling chronic kidney disease in diabetic patients with finerenone. Trends in pharmacological sciences. 2022 Academic Article GET IT
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Magmas Inhibition in Prostate Cancer: A Novel Target for Treatment-Resistant Disease.
Cancers.
2022
Academic Article
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Times cited: 8 -
Potential therapeutic roles of retinoids for prevention of neuroinflammation and neurodegeneration in Alzheimer's disease.
Neural regeneration research.
2019
Review
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Times cited: 75 -
Discovery of a Small Molecule Promoting Mouse and Human Osteoblast Differentiation via Activation of p38 MAPK-β.
Cell chemical biology.
2019
Academic Article
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Times cited: 20 -
The ceramide synthase 2b gene mediates genomic sensing and regulation of sphingosine levels during zebrafish embryogenesis.
eLife.
2017
Academic Article
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Times cited: 22 -
Retinoic acid signaling pathways in development and diseases.
Bioorganic & medicinal chemistry.
2013
Review
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Times cited: 224 -
Use of zebrafish in chemical biology and drug discovery.
Future medicinal chemistry.
2013
Review
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Times cited: 15 -
Boron chemicals in diagnosis and therapeutics.
Future medicinal chemistry.
2013
Review
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Times cited: 230 -
Design and synthesis of 3,5-disubstituted boron-containing 1,2,4-oxadiazoles as potential combretastatin A-4 (CA-4) analogs.
Tetrahedron letters.
2012
Academic Article
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Times cited: 21 -
Design and synthesis of boron containing potential pan-RAR inverse agonists.
Tetrahedron letters.
2012
Academic Article
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Times cited: 9 -
Novel retinoic acid receptor alpha agonists for treatment of kidney disease.
PloS one.
2011
Academic Article
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Times cited: 43 -
Design and Synthesis of 3,5-Disubstituted 1,2,4-Oxadiazole Containing Retinoids from a Retinoic Acid Receptor Agonist.
Tetrahedron letters.
2011
Academic Article
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Times cited: 7 -
Synthesis of function-oriented 2-phenyl-2H-chromene derivatives using L-pipecolinic acid and substituted guanidine organocatalysts.
Tetrahedron letters.
2010
Academic Article
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Times cited: 50 -
A forward chemical screen in zebrafish identifies a retinoic acid derivative with receptor specificity.
PloS one.
2010
Academic Article
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Times cited: 20 -
Design and Synthesis of Potential New Apoptosis Agents: Hybrid Compounds Containing Perillyl Alcohol and New Constrained Retinoids.
Tetrahedron letters.
2010
Academic Article
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Times cited: 17 -
Design and synthesis of novel pinacolylboronate containing combretastatin 'antimitotic agent' analogues.
Tetrahedron letters.
2009
Academic Article
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Times cited: 15 -
Design and synthesis of (E)-1-((3-ethyl-2,4,4-trimethylcyclohex-2-enylidene)methyl-4-substituted benzenes from 1-(2,6,6-trimethylcyclohex-1-enyl)ethanol.
Chemical communications (Cambridge, England).
2009
Academic Article
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Times cited: 12 -
A forward chemical screen using zebrafish embryos with novel 2-substituted 2H-chromene derivatives.
Chemical biology & drug design.
2009
Academic Article
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Times cited: 39 -
Synthesis of 2-substituted 2H-chromenes using potassium vinyltrifluoroborates.
Tetrahedron letters.
2008
Academic Article
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Times cited: 50