Pillarsetty, Naga Vara Kishore

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selected publications

Improved radiosynthesis of ¹²³I-MAPi, an auger theranostic agent. International journal of radiation biology. 2020 Academic Article GET IT
Times cited: 14
A one-pot radiosynthesis of [¹⁸ F]PARPi. Journal of labelled compounds & radiopharmaceuticals. 2020 Academic Article GET IT
Times cited: 6
The epichaperome is a mediator of toxic hippocampal stress and leads to protein connectivity-based dysfunction. Nature communications. 2020 Academic Article GET IT
Times cited: 44
Paradigms for Precision Medicine in Epichaperome Cancer Therapy. Cancer cell. 2019 Academic Article GET IT
Times cited: 44
Leveraging PET to image folate receptor α therapy of an antibody-drug conjugate. EJNMMI research. 2018 Academic Article GET IT
Times cited: 13
TMSOTf assisted synthesis of 2'-deoxy-2'-[18F]fluoro-β-D-arabinofuranosylcytosine ([18F]FAC). PloS one. 2018 Academic Article GET IT
Times cited: 3
Target engagement imaging of PARP inhibitors in small-cell lung cancer. Nature communications. 2018 Academic Article GET IT
Times cited: 71
Pretargeting of internalizing trastuzumab and cetuximab with a ¹⁸F-tetrazine tracer in xenograft models. EJNMMI research. 2017 Academic Article GET IT
Times cited: 66
In Vitro and In Vivo Comparison of Gemcitabine and the Gemcitabine Analog 1-(2'-deoxy-2'-fluoroarabinofuranosyl) Cytosine (FAC) in Human Orthotopic and Genetically Modified Mouse Pancreatic Cancer Models. Molecular imaging and biology. 2017 Academic Article GET IT
Times cited: 13
Repeatability of [⁶⁸Ga]DKFZ11-PSMA PET Scans for Detecting Prostate-specific Membrane Antigen-positive Prostate Cancer. Molecular imaging and biology. 2017 Academic Article GET IT
Times cited: 6
The epichaperome is an integrated chaperome network that facilitates tumour survival. Nature. 2016 Academic Article GET IT
Times cited: 200
Sustained ERK inhibition maximizes responses of BrafV600E thyroid cancers to radioiodine. The Journal of clinical investigation. 2016 Academic Article GET IT
Times cited: 103
Copper-64 labeled liposomes for imaging bone marrow. Nuclear medicine and biology. 2016 Academic Article GET IT
Times cited: 20
Synthesis and evaluation of an (18)F-labeled pyrimidine-pyridine amine for targeting CXCR4 receptors in gliomas. Nuclear medicine and biology. 2016 Academic Article GET IT
Times cited: 12
Tetrahydroprotoberberine alkaloids with dopamine and σ receptor affinity. Bioorganic & medicinal chemistry. 2016 Academic Article GET IT
Times cited: 19
Radiosynthesis of the iodine-124 labeled Hsp90 inhibitor PU-H71. Journal of labelled compounds & radiopharmaceuticals. 2016 Academic Article GET IT
Times cited: 18
(18)F-Based Pretargeted PET Imaging Based on Bioorthogonal Diels-Alder Click Chemistry. Bioconjugate chemistry. 2015 Academic Article GET IT
Times cited: 132
Radioiodinated PARP1 tracers for glioblastoma imaging. EJNMMI research. 2015 Academic Article GET IT
Times cited: 49
Synthesis and evaluation of (18)F-labeled ATP competitive inhibitors of topoisomerase II as probes for imaging topoisomerase II expression. European journal of medicinal chemistry. 2014 Academic Article GET IT
Times cited: 10
Development of a minimal saponin vaccine adjuvant based on QS-21. Nature chemistry. 2014 Academic Article GET IT
Times cited: 73
Building Blocks for the Construction of Bioorthogonally Reactive Peptides via Solid-Phase Peptide Synthesis. ChemistryOpen. 2014 Academic Article GET IT
Times cited: 24
Increased KIT inhibition enhances therapeutic efficacy in gastrointestinal stromal tumor. Clinical cancer research : an official journal of the American Association for Cancer Research. 2014 Academic Article GET IT
Times cited: 46
Influence of free fatty acids on glucose uptake in prostate cancer cells. Nuclear medicine and biology. 2013 Academic Article GET IT
Times cited: 9
(18)F-labeled-bioorthogonal liposomes for in vivo targeting. Bioconjugate chemistry. 2013 Academic Article GET IT
Times cited: 75
Synthesis and evaluation of 18F-labeled benzylguanidine analogs for targeting the human norepinephrine transporter. European journal of nuclear medicine and molecular imaging. 2013 Academic Article GET IT
Times cited: 49
Tumor-specific targeting with modified Sindbis viral vectors: evaluation with optical imaging and positron emission tomography in vivo. Molecular imaging and biology. 2013 Academic Article GET IT
Times cited: 9
Antilipolytic drug boosts glucose metabolism in prostate cancer. Nuclear medicine and biology. 2013 Academic Article GET IT
Times cited: 5
Fluorine-labeled dasatinib nanoformulations as targeted molecular imaging probes in a PDGFB-driven murine glioblastoma model. Neoplasia (New York, N.Y.). 2012 Academic Article GET IT
Times cited: 40
Efficient (18)F-labeling of large 37-amino-acid pHLIP peptide analogues and their biological evaluation. Bioconjugate chemistry. 2012 Academic Article GET IT
Times cited: 61
An improved strategy for the synthesis of [¹⁸F]-labeled arabinofuranosyl nucleosides. Nuclear medicine and biology. 2012 Academic Article GET IT
Times cited: 12
Dosimetry of 18F-labeled tyrosine kinase inhibitor SKI-249380, a dasatinib-tracer for PET imaging. Molecular imaging and biology. 2012 Academic Article GET IT
Times cited: 10
Affinity-based proteomics reveal cancer-specific networks coordinated by Hsp90. Nature chemical biology. 2011 Academic Article GET IT
Times cited: 230
In vivo imaging of Bcr-Abl overexpressing tumors with a radiolabeled imatinib analog as an imaging surrogate for imatinib. Journal of nuclear medicine : official publication, Society of Nuclear Medicine. 2011 Academic Article GET IT
Times cited: 19
Design and synthesis of a bombesin peptide-conjugated tripodal phosphino dithioether ligand topology for the stabilization of the fac-[M(CO)3]+ core (M=(99 m)Tc or Re). Inorganic chemistry. 2011 Academic Article GET IT
Times cited: 15
The synthesis and evaluation of N1-(4-(2-[18F]-fluoroethyl)phenyl)-N8-hydroxyoctanediamide ([18F]-FESAHA), a PET radiotracer designed for the delineation of histone deacetylase expression in cancer. Nuclear medicine and biology. 2011 Academic Article GET IT
Times cited: 15
Optimizing tumor targeting of the lipophilic EGFR-binding radiotracer SKI 243 using a liposomal nanoparticle delivery system. Journal of controlled release : official journal of the Controlled Release Society. 2010 Academic Article GET IT
Times cited: 34
Improved synthesis of 2'-deoxy-2'-[18F]-fluoro-1-beta-D-arabinofuranosyl-5-iodouracil ([18F]-FIAU). Nuclear medicine and biology. 2010 Academic Article GET IT
Times cited: 28
(124)I-iodopyridopyrimidinone for PET of Abl kinase-expressing tumors in vivo. Journal of nuclear medicine : official publication, Society of Nuclear Medicine. 2010 Academic Article GET IT
Times cited: 9
2-18F-Fluoropropionic acid as a PET imaging agent for prostate cancer. Journal of nuclear medicine : official publication, Society of Nuclear Medicine. 2009 Academic Article GET IT
Times cited: 33
Multimodality imaging of TGFbeta signaling in breast cancer metastases. FASEB journal : official publication of the Federation of American Societies for Experimental Biology. 2009 Academic Article GET IT
Times cited: 48
Monitoring the efficacy of adoptively transferred prostate cancer-targeted human T lymphocytes with PET and bioluminescence imaging. Journal of nuclear medicine : official publication, Society of Nuclear Medicine. 2008 Academic Article GET IT
Times cited: 79
A new acycloguanosine-specific supermutant of herpes simplex virus type 1 thymidine kinase suitable for PET imaging and suicide gene therapy for potential use in patients treated with pyrimidine-based cytotoxic drugs. Journal of nuclear medicine : official publication, Society of Nuclear Medicine. 2008 Academic Article GET IT
Times cited: 27
Imaging of HSV-tk Reporter gene expression: comparison between [18F]FEAU, [18F]FFEAU, and other imaging probes. Journal of nuclear medicine : official publication, Society of Nuclear Medicine. 2008 Academic Article GET IT
Times cited: 48
Synthesis and biological evaluation of a fluorine-18 derivative of dasatinib. Journal of medicinal chemistry. 2007 Academic Article GET IT
Times cited: 36
Synthesis and evaluation of [18F] labeled pyrimidine nucleosides for positron emission tomography imaging of herpes simplex virus 1 thymidine kinase gene expression. Journal of medicinal chemistry. 2006 Academic Article GET IT
Times cited: 19
Non-invasive molecular imaging and reporter genes. Central European Journal of Biology. 2006 Article GET IT
Imaging herpes viral thymidine kinase-1 reporter gene expression with a new 18F-labeled probe: 2'-fluoro-2'-deoxy-5-[18F]fluoroethyl-1-beta-d-arabinofuranosyl uracil. Nuclear medicine and biology. 2005 Academic Article GET IT
Times cited: 15
Design, synthesis, and chemistry of sterically nondemanding primary bisphosphines. Journal of the American Chemical Society. 2005 Academic Article GET IT
Times cited: 22
Unprecedented rhodium-mediated catalytic transfer hydrogenation of a phosphonate functionalized olefin in ecofriendly media. Inorganica Chimica Acta. 2004 Article GET IT
Characterization of complexation reactions of mono- and bidentate-hydroxymethyl phosphine ligands with the organometallic 99mTc(I)(OH2)3(CO)3+ synthon. Radiochimica Acta. 2003 Article GET IT
Characterization of supramolecular (H2O)18 water morphology and water-methanol (H2O)15(CH3OH)3 clusters in a novel phosphorus functionalized trimeric amino acid host. Journal of the American Chemical Society. 2003 Academic Article GET IT
Times cited: 249
Syntheses, in vitro and in vivo characterization of a 99mTc-(I)-tricarbonyl-benzylamino-dihydroxymethyl phosphine (NP(2)) chelate. Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine. 2003 Academic Article GET IT
Times cited: 17
In vitro and in vivo antitumor properties of tetrakis((trishydroxy- methyl)phosphine)gold(I) chloride. Journal of medicinal chemistry. 2003 Academic Article GET IT
Times cited: 54
Preclinical tolerance and pharmacokinetic assessment of MU-Gold, a novel chemotherapeutic agent, in laboratory dogs. Veterinary therapeutics : research in applied veterinary medicine. 2003 Academic Article GET IT
Times cited: 5
First examples of azaphosphanes as efficient electron donors in the chemical architecture of thermally stable new nonlinear optical materials. Chemistry of Materials. 2002 Article GET IT
Exceptional kinetic propensity of hydroxymethyl phosphanes toward Rh(III) stabilization in water. Journal of the American Chemical Society. 2002 Academic Article GET IT
Times cited: 30
Synthesis and characterization of (99m)Tc- and (188)Re-complexes with a diamido-dihydroxymethylenephosphine-based bifunctional chelating agent (N(2)P(2)-BFCA). Nuclear medicine and biology. 2002 Academic Article GET IT
Times cited: 15

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Background

education and training

Bs.C., Osmania University (India) 96
Ph.D., University of Missouri 2003
M.Sc., University of Hyderabad (India) 1998

Contact

full name

Naga Vara Kishore Pillarsetty

VIVO Weill Cornell Medical College

Naga Vara Kishore Pillarsetty Professor of Radiochemistry and Radiopharmacy in Radiology

Publications

selected publications

Background

education and training

Contact

full name